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137076-22-3 - 1-Boc-piperidine-4-carboxaldehyde, 97% - 1-Boc-4-formylpiperidine - H52813 - Alfa Aesar

H52813 1-Boc-piperidine-4-carboxaldehyde, 97%

CAS Number

Size Price ($) Quantity Availability
250mg 21.90
1g 65.60
5g 262.00
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1-Boc-piperidine-4-carboxaldehyde, 97%


Chemical Properties

Formula Weight
Air Sensitive
Soluble in methanol.


1-Boc-piperidine-4-carboxaldehyde is used as reactant for synthesis of Pim-1 inhibitors, selective GPR119 agonists for type II diabetes, M-tropic (R5) HIV-1 replication inhibitors, HDAC inhibitors and selective 5-HT6 antagonists. It is also used as reactant for three-component vinylogous Mannich reactions


Air sensitive. Incompatible with oxidizing agents.

Literature References

Yibin Xiang; Bradford Hirth; Gary Asmussen; Hans-Peter Biemann; Kimberly A.Bishop; Andrew Good; Maria Fitzgerald; Tatiana Gladysheva; Annuradha Jain; Katherine Jancsics; Jinyu Liu; Markus Metz; Andrew Papoulis; Renato Skerlj; J.David Stepp; Ronnie R.Wei. The discovery of novel benzofuran-2-carboxylic acids as potent Pim-1 inhibitors. Bioorganic & Medicinal Chemistry Letters. 2011, 21, (10),3050-3056


Jason W.Szewczyk; John Acton; Alan D.Adams; Gary Chicchi; Stanley Freeman; Andrew D.Howard; Yong Huang; Cai Li; Peter T.Meinke; Ralph Mosely; Elizabeth Murphy; Rachel Samuel; Conrad Santini; Meng Yang; Yong Zhang; Kake Zhao; Harold B.Wood. Design of potent and selective GPR119 agonists for type II diabetes. Bioorganic & Medicinal Chemistry Letters. 2011, 21, (9),2665-2669

GHS Hazard and Precautionary Statements

Hazard Statements: H315-H319-H335

Causes skin irritation. Causes serious eye irritation. May cause respiratory irritation.

Precautionary Statements: P261-P280a-P305+P351+P338-P304+P340-P405-P501a

Avoid breathing dust/fume/gas/mist/vapours/spray. Wear protective gloves and eye/face protection. IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continue rinsing. IF INHALED: Remove to fresh air and keep at rest in a position comfortable for breathing. Store locked up. Dispose of contents/container in accordance with local/regional/national/international regulations.

Other References

Harmonized Tariff Code


  • A13697

    Diethyl iodomethylphosphonate, 98+%
  • A14120

    Triethyl phosphonoacetate, 98+%
  • H52571

    1-Boc-piperidine-3-carboxaldehyde, 97%

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